Vassilis J. Demopoulos: search on Z-Library

The world's largest scientific articles store. 70,000,000+ articles for free.

1

Formation of novel N-acetylcysteine-hemin adducts abrogates hemin-induced cytotoxicity and suppresses the NRF2-driven stress response in human pro-erythroid K562â¯cells

Georgiou-Siafis, Sofia K., Samiotaki, Martina K., Demopoulos, Vassilis J., Panayotou, George, Tsiftsoglou, Asterios S.

Journal:

European Journal of Pharmacology

Year:

2020

Language:

english

File:

PDF, 8.33 MB

english, 2020

2

Aldose Reductase Enzyme and its Implication to Major Health Problems of the 21st Century

Alexiou, Polyxeni, Pegklidou, Kyriaki, Chatzopoulou, Maria, Nicolaou, Ioannis, Demopoulos, Vassilis

Journal:

Current Medicinal Chemistry

Year:

2009

Language:

english

File:

PDF, 516 KB

english, 2009

3

Decreasing acidity in a series of aldose reductase inhibitors: 2-Fluoro-4-(1H-pyrrol-1-yl)phenol as a scaffold for improved membrane permeation

Chatzopoulou, Maria, Patsilinakos, Alexandros, Vallianatou, Theodosia, Prnova, Marta Soltesova, Žakelj, Simon, Ragno, Rino, Stefek, Milan, Kristl, Albin, Tsantili-Kakoulidou, Anna, Demopoulos, Vassili

Journal:

Bioorganic & Medicinal Chemistry

Year:

2014

Language:

english

File:

PDF, 1.97 MB

english, 2014

4

Structure–activity relations on [1-(3,5-difluoro-4-hydroxyphenyl)-1H-pyrrol-3-yl]phenylmethanone. The effect of methoxy substitution on aldose reductase inhibitory activity and selectivity

Maria Chatzopoulou, Eduard Mamadou, Maria Juskova, Cathrine Koukoulitsa, Ioannis Nicolaou, Milan Stefek, Vassilis J. Demopoulos

Journal:

Bioorganic & Medicinal Chemistry

Year:

2011

Language:

english

File:

PDF, 666 KB

english, 2011

5

HPLC-based lipophilicity of pyrrolyl-acetic acid ARIs: Relationships with biological activity

Marios Chrysanthakopoulos, Ioannis Nicolaou, Vassilis J. Demopoulos, Anna Tsantili-Kakoulidou

Journal:

Journal of Chromatography B

Year:

2010

Language:

english

File:

PDF, 572 KB

english, 2010

6

Lipophilicity Studies on Pyrrolyl-Acetic Acid Derivatives. Experimental Versus Predicted logP Values in Relationship with Aldose Reductase Inhibitory Activity

Marios Chrysanthakopoulos, Antigoni Koletsou, Ioannis Nicolaou, Vassilis J. Demopoulos, Anna Tsantili-Kakoulidou

Journal:

Molecular Informatics

Year:

2009

Language:

english

File:

PDF, 371 KB

english, 2009

7

Substituted Pyrrol-1-ylacetic Acids That Combine Aldose Reductase Enzyme Inhibitory Activity and Ability To Prevent the Nonenzymatic Irreversible Modification of Proteins from Monosaccharides

Nicolaou, Ioannis, Demopoulos, Vassilis J.

Journal:

Journal of Medicinal Chemistry

Year:

2003

Language:

english

File:

PDF, 332 KB

english, 2003

8

SYNTHESIS OF N-PROTECTED 1 H -INDOLE-5-CARBOXYLIC ACIDS WITH ALDOSE REDUCTASE INHIBITORY POTENTIAL

Nicolaou, Ioannis, Zaher, Nazlaa, Demopoulos, Vassilis J.

Journal:

Organic Preparations and Procedures International

Year:

2002

Language:

english

File:

PDF, 235 KB

english, 2002

9

A CONVENIENT “HYDROGEN TRANSFER” HYDROGENATION OF TESTOSTERONE

Spyriounis, Dimitris M., Ikonomidis, George, Demopoulos, Vassilis J.

Journal:

Organic Preparations and Procedures International

Year:

1989

Language:

english

File:

PDF, 180 KB

english, 1989

10

A CONVENIENT SYNTHESIS OF PYRROLE-3-CARBOXALDEHYDE

Demopoulos, Vassilis J.

Journal:

Organic Preparations and Procedures International

Year:

1986

Language:

english

File:

PDF, 157 KB

english, 1986

11

A Facile Preparation of 1-(6-Hydroxyindol-1-yl)-2,2-dimethylpropan-1-one

Demopoulos, Vassilis John, Nicolaou, Ioannis, Zika, Chariklia

Journal:

CHEMICAL & PHARMACEUTICAL BULLETIN

Year:

2003

Language:

english

File:

PDF, 67 KB

english, 2003

12

A Facile Preparation of 1-(6-Hydroxyindol-1-yl)-2,2-dimethylpropan-1-one.

Vassilis John Demopoulos, Ioannis Nicolaou, Chariklia Zika

Journal:

Year:

2003

File:

PDF, 7 KB

2003

13

Phase Transfer Catalyzed Aromatic Nucleophilic Substituticn of Triflate Esters of 2-and 4-Nitro-estrone

Spyriounis, Dimitris M., Rekka, Eleni, Demopoulos, Vassilis J.

Journal:

Synthetic Communications

Year:

1990

Language:

english

File:

PDF, 313 KB

english, 1990

14

Synthesis of N-Protected 1H-Indole-5-carboxylic Acids (VI) with Aldose Reductase Inhibitory Potential.

Ioannis Nicolaou, Nazlaa Zaher, Vassilis J. Demopoulos

Journal:

Year:

2002

File:

PDF, 27 KB

2002

15

Novel aldose reductase inhibitors: a patent survey (2006 – present)

Chatzopoulou, Maria, Alexiou, Polyxeni, Kotsampasakou, Eleni, Demopoulos, Vassilis J

Journal:

Expert Opinion on Therapeutic Patents

Year:

2012

Language:

english

File:

PDF, 734 KB

english, 2012

16

The AlCL 3 Catalyzed Benzoylation of Ethyl Pyrrole-2-Acetate: An Unusual 6-Substitution

Alexandrou, Elena, Rekka, Eleni, Demopoulos, Vassilis J.

Journal:

Synthetic Communications

Year:

1992

Language:

english

File:

PDF, 256 KB

english, 1992

17

ChemInform Abstract: Clauson-Kaas-Type Synthesis of Pyrrolyl-phenols, from the Hydrochlorides of Aminophenols, in the Presence of Nicotinamide.

Chatzopoulou, Maria, Kotsampasakou, Eleni, Demopoulos, Vassilis J.

Journal:

Year:

2014

File:

PDF, 22 KB

2014

18

Pyrrolylbenzothiazole Derivatives as Aldose Reductase Inhibitors

Zaher, Nazlaa, Nicolaou, Ioannis, Demopoulos, Vassilis J.

Journal:

Journal of Enzyme Inhibition and Medicinal Chemistry

Year:

2002

Language:

english

File:

PDF, 250 KB

english, 2002

19

Kurzmitteilungen: Synthesis and Biological Evaluation of 3-(2-Aminoethyl)pyrrole Derivatives Synthese und biologische Bewertung von 3-(2-Aminoethyl)pyrrol-Derivaten

Vassilis J. Demopoulos, Ekaterini Tani, John Paul Long

Journal:

Archiv der Pharmazie

Year:

1989

Language:

english

File:

PDF, 190 KB

english, 1989

20

Evaluation of aldose reductase inhibition and docking studies of 6′-nitro and 6′,6″-dinitrorosmarinic acids

Catherine Koukoulitsa, Fabrice Bailly, Kiriaki Pegklidou, Vassilis J. Demopoulos, Philippe Cotelle

Journal:

European Journal of Medicinal Chemistry

Year:

2010

Language:

english

File:

PDF, 595 KB

english, 2010

21

Clauson–Kaas-Type Synthesis of Pyrrolyl-phenols, from the Hydrochlorides of Aminophenols, in the Presence of Nicotinamide

Chatzopoulou, Maria, Kotsampasakou, Eleni, Demopoulos, Vassilis J.

Journal:

Synthetic Communications

Year:

2013

Language:

english

File:

PDF, 198 KB

english, 2013

22

Design and synthesis of novel series of pyrrole based chemotypes and their evaluation as selective aldose reductase inhibitors. A case of bioisosterism between a carboxylic acid moiety and that of a tetrazole

Kyriaki Pegklidou, Catherine Koukoulitsa, Ioannis Nicolaou, Vassilis J. Demopoulos

Journal:

Bioorganic & Medicinal Chemistry

Year:

2010

Language:

english

File:

PDF, 1.60 MB

english, 2010

23

ChemInform Abstract: A Study of the Friedel-Crafts Acylation of 1-Benzenesulfonyl-1H-pyrrole in the Preparation of 3-Aroylpyrroles.

Ioannis Nicolaou, Vassilis J. Demopoulos

Journal:

Year:

1999

File:

PDF, 28 KB

1999

24

A study of the friedel-crafts acylation of 1-benzenesulfonyl-1H-pyrrole in the preparation of 3-aroylpyrroles

Ioannis Nicolaou, Vassilis J. Demopoulos

Journal:

Journal of Heterocyclic Chemistry

Year:

1998

File:

PDF, 239 KB

1998

25

Evaluation of aldose reductase inhibition and docking studies of some secondary metabolites, isolated from Origanum vulgare L. ssp. hirtum

Catherine Koukoulitsa, Chariklia Zika, George D. Geromichalos, Vassilis J. Demopoulos, Helen Skaltsa

Journal:

Bioorganic & Medicinal Chemistry

Year:

2006

Language:

english

File:

PDF, 518 KB

english, 2006

26

[1-(3,5-Difluoro-4-hydroxyphenyl)-1 H -pyrrol-3-yl]phenylmethanone as a Bioisostere of a Carboxylic Acid Aldose Reductase Inhibitor

Nicolaou, Ioannis, Zika, Chariklia, Demopoulos, Vassilis J.

Journal:

Journal of Medicinal Chemistry

Year:

2004

Language:

english

File:

PDF, 52 KB

english, 2004

27

A Diverse Series of Substituted Benzenesulfonamides as Aldose Reductase Inhibitors with Antioxidant Activity: Design, Synthesis, and in Vitro Activity

Alexiou, Polyxeni, Demopoulos, Vassilis J.

Journal:

Journal of Medicinal Chemistry

Year:

2010

Language:

english

File:

PDF, 1007 KB

english, 2010

28

Isomeric benzoylpyrroleacetic acids: Some structural aspects for aldose reductase inhibitory and anti-inflammatory activities

Vassilis J. Demopoulos, Eleni Rekka

Journal:

Journal of Pharmaceutical Sciences

Year:

1995

Language:

english

File:

PDF, 452 KB

english, 1995

29

Synthesis of N-acyl-2-pyrrolidinones from the corresponding N-acyl-GABA derivatives

George V. Rekatas, Vassilis J. Demopoulos, Panos N. Kourounakis

Journal:

Journal of Heterocyclic Chemistry

Year:

1996

File:

PDF, 124 KB

1996

30

Bis-pyrrolyl-tetrazolyl derivatives as hybrid polar compounds: A case of lipophilic functional bioisosterism with bis-acetamides

Maria Chatzopoulou, Ioannis D. Bonovolias, Ioannis Nicolaou, Vassilis J. Demopoulos, Ioannis S. Vizirianakis, Asterios S. Tsiftsoglou

Journal:

European Journal of Medicinal Chemistry

Year:

2012

Language:

english

File:

PDF, 446 KB

english, 2012

31

A One-Step Conversion of Certain Indole and Pyrrole Glyoxtlic Acid Esters to the Corresponding Acetates

Demopoulos, Vassilis J.

Journal:

Synthetic Communications

Year:

1989

Language:

english

File:

PDF, 356 KB

english, 1989

32

Cu(II) complex of an estradiol derivative with potent anti-inflammatory properties

Dimitris M. Spyriounis, Eleni Rekka, Vassilis J. Demopoulos, Panos N. Kourounakis

Journal:

Archiv der Pharmazie

Year:

1991

Language:

english

File:

PDF, 341 KB

english, 1991

33

Carboxymethylated pyridoindole antioxidants as aldose reductase inhibitors: Synthesis, activity, partitioning, and molecular modeling

Milan Stefek, Vladimir Snirc, Paul-Omer Djoubissie, Magdalena Majekova, Vassilis Demopoulos, Lucia Rackova, Zelmira Bezakova, Cimen Karasu, Vincenzo Carbone, Ossama El-Kabbani

Journal:

Bioorganic & Medicinal Chemistry

Year:

2008

Language:

english

File:

PDF, 535 KB

english, 2008

34

Design and synthesis of N-(3,5-difluoro-4-hydroxyphenyl)benzenesulfonamides as aldose reductase inhibitors

Polyxeni Alexiou, Ioannis Nicolaou, Milan Stefek, Albin Kristl, Vassilis J. Demopoulos

Journal:

Bioorganic & Medicinal Chemistry

Year:

2008

Language:

english

File:

PDF, 192 KB

english, 2008

35

Inhibitory effect of polar oregano extracts on aldose reductase and soybean lipoxygenase in vitro

Catherine Koukoulitsa, Chariklia Zika, Dimitra Hadjipavlou–Litina, Vassilis J. Demopoulos, Helen Skaltsa

Journal:

Phytotherapy Research

Year:

2006

Language:

english

File:

PDF, 76 KB

english, 2006

36

Lipophilicity of Some Substituted Morpholine Derivatives Synthesized as Potential Antinociceptive Agents

Eleni Rekka, Stavros Retsas, Vassilis J. Demopoulos, Panos N. Kourounakis

Journal:

Archiv der Pharmazie

Year:

1990

Language:

english

File:

PDF, 357 KB

english, 1990

37

Synthesis of 3-(2-Aminoethyl)pyrrole Derivatives

Vassilis J. Demopoulos

Journal:

Journal of Heterocyclic Chemistry

Year:

1988

File:

PDF, 320 KB

1988

38

Fraction Lipophilicity Index (FLI)

Tsantili-Kakoulidou, Anna, Chatzopoulou, Maria, Demopoulos, Vassilis J.

Journal:

International Journal of Quantitative Structure-Property Relationships

Year:

2019

Language:

english

File:

PDF, 1.89 MB

english, 2019

39

Substituted derivatives of indole acetic acid as aldose reductase inhibitors with antioxidant activity: structure-activity relationship

Juskova, Maria, Majekova, Magdalena, Demopoulos, Vassilis, Stefek,  Milan

Journal:

General Physiology and Biophysics

Year:

2012

Language:

english

File:

PDF, 536 KB

english, 2012

40

Synthesis of 6,7,8,9-tetrahydro-N,N-di-n-propyl-1H-benz[g] indol-7-amine, a potential dopamine receptor agonist

Vassilis J. Demopoulos, Antonis Gavalas, George Rekatas, Ekaterini Tani

Journal:

Journal of Heterocyclic Chemistry

Year:

1995

File:

PDF, 320 KB

1995

41

Toward the Development of Innovative Bifunctional Agents To Induce Differentiation and To Promote Apoptosis in Leukemia: Clinical Candidates and Perspectives

Vizirianakis, Ioannis S., Chatzopoulou, Maria, Bonovolias, Ioannis D., Nicolaou, Ioannis, Demopoulos, Vassilis J., Tsiftsoglou, Asterios S.

Journal:

Journal of Medicinal Chemistry

Year:

2010

Language:

english

File:

PDF, 1.71 MB

english, 2010

42

The efficiency of RP-TLC for lipophilicity assessment. A comparative study on a series of pyrrolyl-acetic acid derivatives, inhibitors of aldose reductase

Chrysanthakopoulos, Marios, Nicolaou, Ioannis, Demopoulos, Vassilis, Tsantili-Kakoulidou, Anna

Journal:

JPC - Journal of Planar Chromatography - Modern TLC

Year:

2012

Language:

english

File:

PDF, 160 KB

english, 2012

43

Synthesis of derivatives of the keto-pyrrolyl-difluorophenol scaffold: Some structural aspects for aldose reductase inhibitory activity and selectivity

Kotsampasakou, Eleni, Demopoulos, Vassilis J.

Journal:

Bioorganic & Medicinal Chemistry

Year:

2013

Language:

english

File:

PDF, 272 KB

english, 2013

44

Behavioral and antioxidant activity of a tosylbenz[g]indolamine derivative. A proposed better profile for a potential antipsychotic agent

Chara A Zika, Ioannis Nicolaou, Antonis Gavalas, George V Rekatas, Ekaterini Tani, Vassilis J Demopoulos

Journal:

Annals of General Psychiatry

Year:

2004

Language:

english

File:

PDF, 1.10 MB

english, 2004

45

A Study of the Electrophilic Aroylation of 1-Aryl-1 H -pyrroles: An Improved Preparation of an Active and Selective Aldose Reductase Inhibitor

Kontonikas, Nikolaos, Kotsampasakou, Panagiota, Sakalis, Nikolaos, Demopoulos, Vassilis J.

Journal:

Organic Preparations and Procedures International

Year:

2019

File:

PDF, 576 KB

2019

46

Synthesis of GABA-Valproic Acid Derivatives and Evaluation of Their Anticonvulsant and Antioxidant Activity

George V. Rekatas, Ekaterini Tani, Vassilis J. Demopoulos, Panos N. Kourounakis

Journal:

Archiv der Pharmazie

Year:

1996

Language:

english

File:

PDF, 582 KB

english, 1996

47

A combinatorial access to 1,5-benzodiazepine derivatives and their evaluation for aldose reductase inhibition

Minodora Pozarentzi, Julia Stephanidou-Stephanatou, Constantinos A. Tsoleridis, Chariklia Zika, Vassilis Demopoulos

Journal:

Year:

2009

Language:

english

File:

PDF, 540 KB

english, 2009

48

Development of aldose reductase inhibitors for the treatment of inflammatory disorders

Chatzopoulou, Maria, Pegklidou, Kyriaki, Papastavrou, Nikolaos, Demopoulos, Vassilis J

Journal:

Expert Opinion on Drug Discovery

Year:

2013

Language:

english

File:

PDF, 662 KB

english, 2013

49

Electrophilic Substitution of Indole on the Benzene Moiety: A Synthesis of 5-Acyl- and 5-Aroylindoles

Demopoulos, Vassilis J.

Journal:

Year:

1998

Language:

english

File:

PDF, 37 KB

english, 1998

50

Nutritional Overview on the Management of Type 2 Diabetes and the Prevention of its Complications

Pegklidou, Kyriaki, Nicolaou, Ioannis, J. Demopoulos, Vassilis

Journal:

Current Diabetes Reviews

Year:

2010

Language:

english

File:

PDF, 179 KB

english, 2010

To build up a library is to create a life. It’s never just a random collection of books.

— Carlos María Domínguez

Official channel

Z-Library Desktop Launcher

Z-Library Since 2009 support@1delivery.pm

EnglishРусскийEspañolItalianoελληνικάاللغة العربيةBahasa IndonesiaBahasa Malaysiaहिन्दीDeutschFrançaisPortuguêsУкраїнськаPolski中文繁體中文日本語Tiếng ViệtAzərbaycan DiliՀայոց լեզուภาษาไทยTürk Diliქართველიবাংলাپښتوతెలుగుاردو한국어SrpskiБългарски